99% Tianeptinum sodium sal CAS 30123-17-2
Specification
ITEM | VEXILLUM | RESULT |
Aspectus | Alba ad flavo pulveris | Album pulveris crystallini |
Solubilitas | Sponte solutum in aqua et methanolum et dichloromethane | Conforms |
Lepidium sativum | Per IR, Ut congruit cum operantes vexillum | Conforms |
(II) dat reactionem sodium | Conforms | |
immunditias A | ≤0.1% | Non detectum |
Related composita | Quis Max unum impurity≤0.1% | 0.093% |
Totalis impurities≤0.4% | 0.36% | |
RELICTUM Solvents (GC) | Acetidin≤ 0.5% | ND |
Dichloromethane≤ 0.06% | ND | |
Methanol≤ 0.3% | ND | |
Acetone≤ 0.5% | 0.29% | |
Acetonitrile≤0.041% | 0.122% | |
Ethanol≤0.5% | ND | |
N, N-dimethylformamide≤0.088% | ND | |
Aquae | ≤ 5.0% | 3.8% |
Temptare (HPLC) | 99.0%-101.0%(On anhydrousbasis) | 99.70% |
Applicationem
Sodium Tianeptinesaltricyclica antidepressant est.Eius mechanismus antidepressans differt ab antidepressantibus tricyclicis traditis.Augere potest restitutionem 5-HT in fissura synaptico.Effectus conductionis HT neuronal.Nulla affinitas cum receptoribus cholini vel adrenergicis.Efficacia antidepressans tricyclicis similis est, tolerabilitas autem melior quam tricyclicorum.Ad curationem tristitiae lenis, moderatae vel graves, tristitia neurogenica et reactiva, anxietas et depressio corporis, praesertim gastrointestinae molestiae, et anxietas et demissio aegrorum alcoholi-dependentium in recessu.